Patent · US Expired

Oxadiazolylimidazobenzodiazepine, compositions, and method

US4622320A · kind A · utility

5Cited by
3References
6Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJan 6, 1986
Grant dateNov 11, 1986
Priority date
Expiry dateJan 6, 2006

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D487/14
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The application discloses novel benzodiazepine agonist compounds, namely, 3-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-5,6-dihydro-5-methyl-6-oxo-7-halo-4 H-imidazo [1,5-a][1,4]benzodiazepines, pharmaceutical compositions thereof, and a method of ameliorating central nervous system ailments therewith, especially convulsions and anxiolytic states. A novel intermediate and process for their production are also disclosed.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.