Aromatic basic-tailed vasopressin antagonists
US4624943A · kind A · utility
1Cited by
3References
16Claims
0Family size
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Key dates
| Filing date | Mar 20, 1985 |
| Grant date | Nov 25, 1986 |
| Priority date | — |
| Expiry date | Mar 20, 2005 |
Classification
- Technology area (CPC Y)Emerging Cross-Sectional Technologies
- CPC primaryY10S930/15
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
Certain new vasopressin-like peptides which have structures characterized by having a bisaminoalkylbenzene present in the vasopressin tail at the 7- or 8-position retain vasopressin antagonist activity. A species of the invention is [1-.beta.-mercapto-.beta.,.beta.-cyclopentamethylenepropionic acid)-2-(O-ethyl)-D-tyrosine-4-valine-8-1',4'-bis(aminomethyl)benzene-9-de sglycinamide]-vasopressin.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.