Patent · US Expired

Aralykyl (arylethynyl)aralkyl amines and their use as vasodilators and antihypertensives

US4661635A · kind A · utility

15Cited by
1References
32Claims
0Family size

Assignee

Inventor

Key dates

Filing dateOct 29, 1984
Grant dateApr 28, 1987
Priority date
Expiry dateOct 29, 2004

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07F1/08
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Acetylenes of the formula (I): ##STR1## wherein Y, m, R.sup.1, R.sup.2 q, Alk, R.sup.3, n and R.sup.4 are as defined herein and Ar.sup.1 and Ar.sup.2 are aromatic, including the salts and ammonium derivatives of formula (I), in treating angina, hypertension and cardiac arrhythmias. Pharmaceutical compositions, methods of use and synthesis and novel intermediates are also part of the invention.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.