Patent · US Expired

Preparation of solid medicament formulation containing nitrendipine

US4724141A · kind A · utility

15Cited by
3References
3Claims
0Family size

Assignee

Inventors

Key dates

Filing dateSep 5, 1985
Grant dateFeb 9, 1988
Priority date
Expiry dateSep 5, 2005

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K31/44
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

A solid medicament formulation comprising 1 part by weight of crystalline nitrendipine, 0.5-1 part by weight of polyvinylpyrrolidone, 0.05-0.5 part by weight of sodium lauryl-sulphate, 1-6 parts by weight of corn starch, 0.5-4 parts by weight of microcrystalline cellulose, 0-5 parts by weight of lactose and 0.01-0.05 parts by weight of magnesium stearate. Such small size formulation has a high bioavailability.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.