Patent · US Expired

Oxadiazolylimidazobenzodiazepine, compositions, and method III

US4745112A · kind A · utility

2Cited by
4References
6Claims
0Family size

Assignee

Inventors

Key dates

Filing dateApr 28, 1986
Grant dateMay 17, 1988
Priority date
Expiry dateApr 28, 2006

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D487/14
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The application discloses novel benzodiazepine agonist compounds, namely, compounds having the formula ##STR1## wherein X is F, CF.sub.3, CH.sub.3, or CN, pharmaceutical compositions thereof, and a method of ameliorating central nervous system ailments therewith, especially convulsions and anxiolytic states. A novel intermediate and process for their production are also disclosed.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.