Assay for D-1 antagonistic activity of neuroleptic drugs
US4760029A · kind A · utility
3Cited by
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Key dates
| Filing date | Nov 19, 1984 |
| Grant date | Jul 26, 1988 |
| Priority date | — |
| Expiry date | Nov 19, 2004 |
Classification
- Technology area (CPC Y)Emerging Cross-Sectional Technologies
- CPC primaryY10S436/815
- WIPO fieldMeasurement
- WIPO sectorInstruments
Abstract
A method, reagents, and kit for determining the levels of D-1 receptor antagonistic activity of neuroleptic drugs. The method correlates competition between analyte and tritiated R-(+)-8-chloro-2,3,4,5-tetrahydro-3-methyl-5-phenyl-1H-3-benzazepin-7-ol for binding to D-1 receptors in mammalian brain tissue.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.