N-indolylethyl-sulphonic acid amides and their use

US4774240A · kind A · utility

Assignee

• BAYER HEALTHCARE LLC · DE

Inventors

• Horst Boshagen · Haan, DE
• Ulrich Rosentreter · Binnen, DE
• Folker Lieb · Leverkusen, DE
• Hermann Oediger · Cologne, DE
• Friedel Seuter
• Elisabeth Perzborn · Wuppertal, DE
• Volker-Bernd Fiedler · Leverkusen, DE

Key dates

• Filing date: Apr 14, 1986
• Grant date: Sep 27, 1988
• Expiry date: Apr 14, 2006

Classification

• Technology area (CPC C): Chemistry; Metallurgy
• CPC primary: C07D417/12
• WIPO field: Organic fine chemistry
• WIPO sector: Chemistry

Abstract

The invention relates to N-indolylethyl-sulphonic acid amides of the formula ##STR1## wherein R.sup.1, R.sup.2, R.sup.3, R.sup.4 and R.sup.5 are defined in the specification and X is carboxyl, alkoxycarbonyl, cyano or carboxamido. These active compounds are useful in medicaments in combating thromboses, thromboembolisms, allergies or asthmatic disorders.