Patent · US Expired

Dihydropyridine anti-allergic and anti-inflammatory agents

US4801598A · kind A · utility

5Cited by
1References
14Claims
0Family size

Assignee

Inventors

Key dates

Filing dateOct 30, 1987
Grant dateJan 31, 1989
Priority date
Expiry dateOct 30, 2007

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D417/14
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Compounds of the formula: ##STR1## where R is 2-substituted phenyl said substituent being chloro, bromo, cyano, methyl, methylthio, methylsulfonyl, trifluoromethyl, hydroxy, methoxy or benzyloxy; R.sup.1 is hydrogen, lower alkyl, pyridyl, thiazolyl, isoxazolyl, thiadiazdyl or thiazdylmethyl; R.sup.2 is hydrogen or lower alkyl; R.sup.3 is hydroxy, lower alkoxy, benzyloxy, amino, lower alkylamino or morpholino; Y is alkylene having two to six carbon atoms; and X is benzimidazolyl optionally substituted by lower alkyl, chloro or trifluoromethyl.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.