Patent · US Expired

Pyrazole-3-amines as anti-inflammatory agents

US4803216A · kind A · utility

18Cited by
0References
10Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 5, 1987
Grant dateFeb 7, 1989
Priority date
Expiry dateMay 5, 2007

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D231/38
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

There are described compounds of formula I, ##STR1## in which R.sub.1 represents hydrogen, alkyl, alkanoyl or alkyl substituted by Ar.sub.1, PA0 R.sub.3, R.sub.4 and R.sub.5, which may be the same or different, each independently represent hydrogen, alkyl or Ar.sub.3, PA0 Ar.sub.1, Ar.sub.2 and Ar.sub.3, which may be the same or different, independently represent phenyl or phenyl substituted by one or more of alkyl, hydroxy, alkoxy, NR.sub.6 R.sub.7 or halogen, PA0 R.sub.6 and R.sub.7, which may be the same or different, independently represent hydrogen or alkyl, and pharmaceutically acceptable acid addition salts thereof. Compositions containing the compounds and methods for their preparation are also described. The compounds are indicated for use as pharmaceutical, e.g. anti-inflammatory, agents.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.