Patent · US Expired

Tetrahydro carbazolone intermediates

US4822881A · kind A · utility

13Cited by
6References
2Claims
0Family size

Assignee

Inventors

Key dates

Filing dateNov 27, 1987
Grant dateApr 18, 1989
Priority date
Expiry dateNov 27, 2007

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D403/06
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The invention relates to compounds of the general formula (I): ##STR1## wherein Im represents an imidazolyl group of the formula: ##STR2## and the various substituents are defined hereinbelow. The compounds are potent and selective antagonists of the effect of 5-HT at 5-HT.sub.3 receptors and are useful, for example, in the treatment of psychotic disorders, anxiety, and nausea and vomiting.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.