Patent · US Expired

Derivatives of pyridoindole, having anti-tumor properties

US4835160A · kind A · utility

11Cited by
0References
13Claims
0Family size

Assignees

Inventors

Key dates

Filing dateMar 17, 1987
Grant dateMay 30, 1989
Priority date
Expiry dateMar 17, 2007

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D471/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention concerns derivatives of 5H-pyrido[4,3-b]-indole with the following general formula: ##STR1## in which n represents a whole number from 2 to 4, R.sub.1 represents hydrogen or a lower alkyl group; R.sub.2 represents hydrogen, a hydroxy group or a lower alkyloxy group; R.sub.3 and R.sub.4 represents hydrogen, a lower alkyl group or hydroxyalkyl group, R.sub.5 can be identical or different and represents hydrogen, a hydroxy group or a lower alkyl group, as well as the tautomeric forms and the addition salts with pharmaceutically acceptable mineral or organic acids. The invention also concerns their preparation process, and their use as medicaments.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.