Patent · US Expired

Isocoumarins with basic substituents as serine proteases inhibitors, anticoagulants and anti-inflammatory agents

US4845242A · kind A · utility

36Cited by
1References
3Claims
0Family size

Assignee

Inventors

Key dates

Filing dateApr 28, 1987
Grant dateJul 4, 1989
Priority date
Expiry dateApr 28, 2007

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D311/76
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Substituted isocoumarins, their preparation, their use in inhibiting serine proteases with trypsin-like, chymotrypsin-like and elastase-like specificity and their roles as anticoagulant agents, and anti-inflammatory agents.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.