Patent · US Expired

Process for the preparation of a 4,5-tri or tetramethylene-4-isothiazoline-3-one

US4851541A · kind A · utility

8Cited by
7References
3Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJun 5, 1986
Grant dateJul 25, 1989
Priority date
Expiry dateJun 5, 2006

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P31/10
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

A process for preparing a 4,5-tri or tetramethylene-4-isothiazoline-3-one comprises cyclizing a 2-alkyl or aralkyl thio-1-cycloalkene-1-carboxamide in the form of its sulfoxide in an organic solvent in the presence of a acid chloride and adding to the resulting 4,5-tri or tetramethylene-4-isothiazoline-3-one hydrochloride a mineral or organic base or water so as to free the 4,5-tri or tetramethylene-4-isothiazoline-3-one in the form of a free base.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.