Patent · US Expired

Antihistaminic benzimidazole derivatives

US4857536A · kind A · utility

2Cited by
1References
5Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJul 22, 1988
Grant dateAug 15, 1989
Priority date
Expiry dateJul 22, 2008

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P37/08
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

A compound which is a benzimidazole derivative of formula (I) ##STR1## in which: R.sub.1 is hydrogen or methyl, PA1 R.sub.2 is hydrogen, methyl or acetyl, PA1 R.sub.3 is hydrogen, methyl or acetyl, and PA1 R.sub.4 is hydrogen or a halogen, PA1 or a pharmaceutically acceptable acid addition salt thereof. The compounds have histamine antagonist activity and are also synthesis intermediates.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.