Patent · US Expired

Noradamantyl-carboxylic acid piperazinoalkyl esters

US4873331A · kind A · utility

26Cited by
1References
6Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 9, 1988
Grant dateOct 10, 1989
Priority date
Expiry dateDec 9, 2008

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D295/088
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The compounds of the following structural formula posses useful anxiolytic, antidepressant, antipsychotic and learning and memory enhancement properties: ##STR1## in which R.sup.1 is 3-noradamantyl; PA1 n is 0 or 1; PA1 X is --CO.sub.2 --, --O.sub.2 C-- or --OCO.sub.2 --; PA1 m is 1, 2, 3, 4, or 5; and PA1 R.sup.2 is phenyl, benzyl, pyridinyl, pyrimidinyl, pyrazinyl or substituted phenyl or benzyl in which the substituent is alkyl, alkoxy, halo, cyano, nitro or trifluoromethyl; or a pharmaceutically acceptable salt thereof.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.