Patent · US Expired

(3S-4S)-7-hydroxy-.DELTA..sup.6 -tetrahydrocannabinols

US4876276A · kind A · utility

53Cited by
5References
10Claims
0Family size

Assignee

Inventors

Key dates

Filing dateOct 26, 1987
Grant dateOct 24, 1989
Priority date
Expiry dateOct 26, 2007

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D311/80
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The invention relates to novel (3S,4S)-7-hydroxy-.DELTA..sup.6 -tetrahydrocannabinol homologes and derivatives, essentially free of the (3R,4R) form and to pharmaceutical compositions which have a potent analgetic, antiemetic and antiglaucoma effect, which compositions contain an effective dosage of a compound of this type. The novel pharmaceutical compositions are practically devoid of the undesired side effects of the (3R,4R) type compounds, such as cannabimimetic psychotropic effects. The pharmaceutical compositions are of special utility in cases of acute and of chronic pain. The invention also relates to a process for the production of the above defined novel compounds.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.