Patent · US Expired

Avermectin derivatives

US4895837A · kind A · utility

21Cited by
3References
15Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJan 13, 1989
Grant dateJan 23, 1990
Priority date
Expiry dateJan 13, 2009

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P33/10
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

There are disclosed novel avermectin .DELTA. 23,24-derivatives (also referred to as 23,24-dehydro compounds). The compounds are prepared by selective dehydration of avermectin A2 or B2 compounds. The avermectin compounds have utility as anti-parasitic agents and compositions for that use are also disclosed. The compounds are also highly potent insecticides against agricultural pests. The .DELTA. 23,24-avermectin compounds have increased activity relative to the A2 or B2 compounds.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.