Patent · US Expired

Aromatic derivatives, their preparation and their use as antimicrobial agents

US4916156A · kind A · utility

9Cited by
5References
12Claims
0Family size

Assignee

Inventors

Key dates

Filing dateApr 6, 1988
Grant dateApr 10, 1990
Priority date
Expiry dateApr 6, 2008

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D233/54
  • WIPO fieldBasic materials chemistry
  • WIPO sectorChemistry

Abstract

The present invention relates to aromatic derivatives of the formula: ##STR1## in which: n represents an integer between 2 and 10; PA1 R.sub.1 and R.sub.2 are identical or different and represent a cycloalkyl containing 3 to 6 carbon atoms or an alkyl containing from 1 to 6 carbon atoms which is unsubstituted or substituted by a phenyl or benzyl group; or PA1 R.sub.1 and R.sub.2, together with the nitrogen atom to which they are bonded, form a heterocycle selected from pyrrolidin-1-yl, piperidino, azepin-1-yl, hexamethyleneimino, 4-methylpiperidino, 4-benzylpiperidino, 4-phenylpiperidino, 1,2,3,4-tetrahydroisoquinol-2-yl, morpholino and imidazol-1-yl groups; PA1 R.sub.3 represents a hydrogen, a halogen, a methyl or a phenyl; PA1 R.sub.4 represents a hydrogen, a halogen or a methyl; or R.sub.3 and R.sub.4, taken together with the benzene ring to which they are bonded, form a naphth-1-yl or naphth-2-yl group; PA1 Y represents a direct bond, a methyleneoxy group, a methylenethio group or a vinylene group; and PA1 R.sub.5 represents an alkyl containing from 5 to 18 carbon atoms, a cycloalkyl containing from 3 to 8 carbon atoms, an adamantyl, naphth-1-yl or naphth-2-yl group, an unsubst…

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.