Substituted azolylmethyl-cyclopropyl-carbinol derivatives

US4921528A · kind A · utility

Assignee

• BAYER HEALTHCARE LLC · DE

Inventors

• Klaus Bockmann · Cologne, DE
• Erik Regel
• Karl H. Buchel · Burscheid, DE
• Klaus Lurssen · Wittlich, DE
• Jorg Konze
• Wilhelm Brandes · Leichlingen, DE

Key dates

• Filing date: Oct 19, 1988
• Grant date: May 1, 1990
• Expiry date: Oct 19, 2008

Classification

• Technology area (CPC C): Chemistry; Metallurgy
• CPC primary: C07D303/36
• WIPO field: Organic fine chemistry
• WIPO sector: Chemistry

Abstract

Plant growth-regulating and fungicidal compounds of the formula ##STR1## in which Ar represents optionally substituted aryl or optionally substituted heteroaryl, PA0 R.sup.1 represents hydrogen, alkyl, alkenyl, alkynyl, trialkylsilyl, optionally substituted phenylalkyl or an acyl radical, PA0 R.sup.2 represents halogen, cyano, thiocyano, alkylcarbonyloxy, alkylcarbonylthio or the groupings --X--R.sup.3 and --NR.sup.4 R.sup.5, PA0 R.sup.3 represents alkyl, cycloalkyl, alkenyl, alkynyl, hydroxyalkyl, alkylthioalkyl, carboxyalkyl, alkoxycarbonylalkyl, optionally substituted aryl, optionally substituted aralkyl or the radical of the formula ##STR2## R.sup.4 and R.sup.3 independently of one another represent hydrogen or alkyl, or PA0 R.sup.4 and R.sup.5, together with the nitrogen atom to which they are bonded, represent an optionally substituted cycloaliphatic ring which can contain further heteroatoms, PA0 X represents oxygen, sulphur, an SO group or an SO.sub.2 group, or PA1 R.sup.2 furthermore represents hydrogen when Ar represents optionally substituted heteroaryl, and PA1 Y represents nitrogen or a CH group, or addition products thereof with acids or metal salts. Novel intermediat…