Patent · US Expired

Platinum complexes with one radiosensitizing ligand

US4921963A · kind A · utility

37Cited by
4References
13Claims
0Family size

Assignee

Inventors

Key dates

Filing dateApr 13, 1987
Grant dateMay 1, 1990
Priority date
Expiry dateApr 13, 2007

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P35/00
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Complexes of platinum II containing a single radiosensitizer ligand and an amino or ammine substituent shows superior binding to DNA and are useful in chemotherapy and sensitization of hypoxic tumors to radiation. The chemotherapeutic value of these compounds is enhanced by administration of vasoactive agents.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.