Patent · US Expired

Novel C.25 (substituted (2-propenyl))-milbemycins

US4927847A · kind A · utility

1Cited by
1References
6Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJul 18, 1989
Grant dateMay 22, 1990
Priority date
Expiry dateJul 18, 2009

Classification

  • Technology area (CPC Y)Emerging Cross-Sectional Technologies
  • CPC primaryY10S435/886
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Antiparasitic milbemycin derivatives having at the C.25 position a substituted 2-propenyl group --C(CH.sub.3).dbd.CH--R.sup.2 wherein R.sup.2 is a C.sub.3 -C.sub.8 alkyl, alkenyl or alkynyl group which may optionally contain an oxygen or sulphur atom as part of the chain, or a C.sub.3 -C.sub.8 cycloalkyl or cycloalkenyl group, or a 3 to 6 membered oxygen or sulphur containing heterocyclic ring which may optionally be substituted by one or more alkyl groups or halogen atoms; and process for their preparation.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.