Patent · US Expired

Smooth muscle cell growth inhibitor

US4945086A · kind A · utility

50Cited by
5References
29Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 3, 1988
Grant dateJul 31, 1990
Priority date
Expiry dateMay 3, 2008

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K38/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

An epithelium-derived inhibitor of the growth of smooth muscle cells is disclosed along with methods for purifying this substance. As initially isolated, the inhibitor comprises a heparan sulfate proteoglycan having a buoyant density of less than 1.4 g/ml which releases a glycosaminoglycan chain having a molecular weight of about 55,000 to 75,000 on protease cleavage. Growth inhibiting activity is found in the glycosaminoglycan chain and in glycosaminoglycan fragments derived therefrom. Use of a dialyzable detergent in purification steps greatly aids in the handling and purification of the inhibitor. The inhibitor can be used in a variety of techniques for inhibiting the growth of smooth muscle cells, both in vivo and in vitro.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.