Patent · US Expired

Cephem compound and a process for preparation thereof

US4952578A · kind A · utility

23Cited by
1References
8Claims
0Family size

Assignee

Inventors

Key dates

Filing dateSep 7, 1988
Grant dateAug 28, 1990
Priority date
Expiry dateSep 7, 2008

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P31/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The object of the invention is a new cephem compound with antimicrobial activity used for the treatment of infectious diseases of the general formula: ##STR1## wherein R1 is amino or a protected amino PA0 R2 is lower alkyl which may have 1 to 3 halogens PA0 R3 is COO.sup..crclbar., carboxy or a protected carboxy PA0 R4 is hydroxy(lower)alkyl or protected hydroxy(lower)alkyl PA0 R5 is amino or a protected amino PA0 R6 is hydrogen or lower alkyl PA0 X.sup..crclbar. is an anion, and PA0 n is 0 or 1 with proviso that PA0 (i) when R3 is COO.sup..crclbar., then n is 0, and PA0 (ii) when R3 is carboxy or a protected carboxy, then n is 1, and pharmaceutically acceptable salt thereof.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.