Patent · US Expired

N-[[6 -methoxy-5-(trifluoromethyl)-1-naphthalenyl]-thioxomethyl]-N-methylglycin e S-oxide and the amide thereof

US4994381A · kind A · utility

1Cited by
13References
1Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMar 20, 1989
Grant dateFeb 19, 1991
Priority date
Expiry dateMar 20, 2009

Classification

  • Technology area (CPC Y)Emerging Cross-Sectional Technologies
  • CPC primaryY10S435/897
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Disclosed herein are N-[[6-methoxy-5-(trifluoromethyl)-1-naphthalenyl]-thioxmethyl]-N-methylgly cine S-oxide (tolrestat S-oxide) and the amine thereof and methods of their preparation. The S-oxides are new aldose reductase inhibitors useful for the treatment or prevention of diabetic complications.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.