Patent · US Expired

New thymopentin retro-inverso analogs and fragments thereof, a process of preparation of the new compounds and the intermediates obtained therein

US5013723A · kind A · utility

8Cited by
3References
5Claims
0Family size

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Inventors

Key dates

Filing dateMar 15, 1988
Grant dateMay 7, 1991
Priority date
Expiry dateMar 15, 2008

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P37/00
  • WIPO fieldBiotechnology
  • WIPO sectorChemistry

Abstract

New retro-inverso analogs of thymopentin (TP5) and of its tripeptide fragment (TP5.sup.1-3) of general formula (I) ##STR1## are described wherein R is hydrogen or an acyl radical, and R.sup.1 is --OR.sup.2 or ##STR2## wherein R.sup.2 is hydrogen or a hydrocarbyl radical, and the corresponding pharmaceutically acceptable acid- or base-addition salts. The new compounds are enzyme-resistant immunomodulatory peptides.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.