Patent · US Expired

Dibenzoheterocyclic hydroxamic acids and hydroxy ureas as inhibitors of 5-lipoxygenase

US5036067A · kind A · utility

12Cited by
10References
9Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMar 14, 1990
Grant dateJul 30, 1991
Priority date
Expiry dateMar 14, 2010

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D337/12
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Compounds having the formula I: ##STR1## are inhibitors of the 5-lipoxygenase enzyme. These compounds are useful as anti-asthmatic, anti-allergic, anti-inflammatory, and cytoprotective agents. They are also useful in treating diarrhea, hypertension, angina, platelet aggregation, cerebral spasm, premature labor, spontaneous abortion, dysmenorrhea, and migraine.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.