Patent · US Expired

Azolyl-derivatives endowed with antifungal activity

US5036094A · kind A · utility

0Cited by
5References
6Claims
0Family size

Assignee

Inventors

Key dates

Filing dateSep 18, 1989
Grant dateJul 30, 1991
Priority date
Expiry dateSep 18, 2009

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D317/22
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Disclosed are compounds, having the general formula: ##STR1## wherein: m=0, 1, 2; n=0, 1 with the condition that when m=0, also n=0; PA0 p=0, 1; q=1, 2; PA0 X is either oxygen or sulphur; PA0 A=N, CH; PA0 R is H, CH.sub.3, F; PA0 R.sub.1 is selected from chlorine, bromine, fluorine, CF.sub.3, phe=nyl, C.sub.1 -C.sub.2 -alkoxy, C.sub.1 -C.sub.2 -haloalkoxy, alkylthio, haloalkyl=thio, wherein the halogen is Cl, Br, F; PA0 R.sub.2 is selected from H, chlorine, bromine, fluorine; PA0 R.sub.f is selected from the group formed by alkyls containing from 2 to 4 carbon atoms, and containing at least 4 atoms of halogen selected from F, Cl and Br, of which at least 3 are F atoms; alkenyls and alkynyls containing up to 4 carbon atoms, containing at least 2 F atoms and, optionally, other halogens selected between Cl and Br. The present invention relates to azolyl-derivatives, more particularly to substituted azolyldioxanes and azolyldioxolanes, endowed with high fungicidal activity, to the process for their preparation, and to their related use in the agrarian field.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.