Derivatives of 1,4-dideoxy-1,4-imino-D-mannitol and preparation thereof
US5041555A · kind A · utility
6Cited by
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4Claims
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Key dates
| Filing date | Sep 21, 1990 |
| Grant date | Aug 20, 1991 |
| Priority date | — |
| Expiry date | Sep 21, 2010 |
Classification
- Technology area (CPC Y)Emerging Cross-Sectional Technologies
- CPC primaryY02P20/582
- WIPO fieldOrganic fine chemistry
- WIPO sectorChemistry
Abstract
Novel derivatives of 1,4-dideoxy-1,4-imino-D-mannitol and method for their synthesis from 4,5-anhydro-1-azido-1-deoxy-2,3-O-isopropylidene-D-talitol or its triflate derivative are disclosed. The novel derivatives, 6-fluoro-1,4-imino-1,4,6-trideoxy-D-mannitol and the N-butyl and N-benzyl derivatives of 1,4-dideoxy-1,4-imino-D-mannitol, have useful mannosidase inhibitory activity.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.