Patent · US Expired

Process for the O-alkylation of N-(hydroxy)aralkylphenylethanolamines

US5041606A · kind A · utility

0Cited by
6References
10Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMar 5, 1990
Grant dateAug 20, 1991
Priority date
Expiry dateMar 5, 2010

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07C2602/10
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

A process for the preparation of a compound of formula ##STR1## wherein X represents hydrogen, halogen, trifluoromethyl or lower alkyl group; W represents methyl, Q represents hydrogen or W and Q, together, form an ethylene group and R' represents a lower alkyl group which comprises protecting the amino group of the phenol corresponding to the compound of formula I, submitting the compound thus obtained to an alkylation (with a compound of formula Hal--CH.sub.2 --COOR', wherein R' is as defined hereinabove for the formula I and Hal is chlorine, bromine or iodine) and then releasing the amino group of the product thus obtained.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.