2-amino-4 or 5-methoxycyclohexyl amides useful as analgesics
US5051428A · kind A · utility
23Cited by
13References
6Claims
0Family size
Assignee
Inventors
Key dates
| Filing date | Mar 29, 1990 |
| Grant date | Sep 24, 1991 |
| Priority date | — |
| Expiry date | Mar 29, 2010 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D333/54
- WIPO fieldOrganic fine chemistry
- WIPO sectorChemistry
Abstract
The invention concerns a series of novel 2-amino-monomethoxycyclohexyl amides having analgesic and neuroprotective activity. The compounds bind selectivity to the kappa opioid receptor. Pharmaceutical compositions containing the compounds, methods of using them, and processes for preparing them are also disclosed.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.