Patent · US Expired

Hexitol derivatives having vasodilative activity

US5053408A · kind A · utility

1Cited by
0References
26Claims
0Family size

Assignee

Inventors

Key dates

Filing dateApr 13, 1990
Grant dateOct 1, 1991
Priority date
Expiry dateApr 13, 2010

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P9/10
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Disclosed is a hexitol derivative represented by the formula (I): ##STR1## wherein Q represents a formula selected from the group consisting of ##STR2## wherein a represents NH, O or S; PA0 each of b, c and d independently represents CH or N; PA0 each of R.sup.1, R.sup.2, R.sup.3 and R.sup.4 independently represents hydrogen, lower alkyl, trifluoromethyl, aryl, lower alkanoyloxy, amino, lower alkylamino, lower alkanoylamino, lower alkanoyl, aroyl, halogen, nitro, (CH.sub.2).sub.m OR.sup. 7, (CH.sub.2).sub.m SR.sup.7, (CH.sub.2).sub.m CO.sub.2 R.sup.7 where R.sup.7 represents hydrogen or lower alkyl and m represents an integer of 0 to 3; PA0 each of R.sup.5 and R.sup.6 independently represents hydrogen or lower alkyl; PA0 U represents >N-- or ##STR3## W represents a single bond, --O-- or --S--; X represents ##STR4## wherein each of Y.sup.1 and Y.sup.2 independently represents hydrogen, lower alkyl, hydroxyl, lower alkanoyloxy, nitrile or phenyl; or Y.sup.1 and Y.sup.2 are combined together to form oxygen; PA0 each of Y.sup.3 and Y.sup.4 independently represents hydrogen or lower alkyl; and l is an integer of 0 to 6, and where l is an integer of 2 to 6, each ##STR5## may be the same …

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.