Phenethylamine derivative compositions and use
US5063246A · kind A · utility
8Cited by
8References
5Claims
0Family size
Assignee
Inventors
Key dates
| Filing date | Aug 21, 1990 |
| Grant date | Nov 5, 1991 |
| Priority date | — |
| Expiry date | Aug 21, 2010 |
Classification
- Technology area (CPC A)Human Necessities
- CPC primaryA61K31/255
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
Phenethylamine derivatives shown by the general formula ##STR1## wherein Ro represents a lower alkyl group; R.sub.1 represents a lower alkyl group or a lower alkoxy group, R.sub.2 represents hydrogen atom or a hydroxyl group; R.sub.3 and R.sub.4 each represents hydrogen atom or a lower alkyl group; R.sub.5 represents hydrogen atom or a lower alkoxy group; X represents oxygen atom or a methylene group; m is an integer of 1-3; and n is an integer of 0-2 and the acid addition salts thereof. These compounds exhibit a strong .alpha.-adrenergic blocking action and are useful as an antihypertensive agent.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.