Patent · US Expired

Process for certain (2R-trans)hexahydroaroquinolizines

US5064964A · kind A · utility

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2References
2Claims
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Assignee

Inventors

Key dates

Filing dateApr 9, 1990
Grant dateNov 12, 1991
Priority date
Expiry dateApr 9, 2010

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D495/22
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

A unique process for preparing certain (2R-trans)hexahydroaroquinolizines, especially (2R-trans)-N-[2-(1,3,4,6,7,12b-hexahydro-2'-oxospiro[aro-[2,3-a]-quinolizi ne-2,4'-imidazolidin]-3'-yl) ethyl)-methanesulfonamide from (2R-trans)-N-[2-[(2-cyano-(1,3,4,6,7,12b-hexahydro-aro-[2,3-a]quinolizin-2 -yl)amino]ethyl]methanesulfonamide is described.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.