Novel benzopyranylpyrrolinone derivatives
US5072006A · kind A · utility
Assignee
Inventors
Key dates
| Filing date | Dec 19, 1990 |
| Grant date | Dec 10, 1991 |
| Priority date | — |
| Expiry date | Dec 19, 2010 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D311/70
- WIPO fieldOrganic fine chemistry
- WIPO sectorChemistry
Abstract
Compounds of the formula ##STR1## wherein: R.sub.1 is cyano or nitro; PA1 R.sub.2 and R.sub.3 are independently hydrogen or lower alkyl; and PA1 R.sub.4 is alkyl; alkenyl; optionally substituted phenyl or phenyl lower alkyl; --(CH.sub.2).sub.m OR.sub.2 or --(CH.sub.2).sub.m N(R.sub.2).sub.2 ; wherein m is an integer of 1-5 and R.sub.2 is as defined above; PA1 or a pharmaceutically acceptable ester thereof; are smooth muscle relaxants, particularly useful in the treatment of hypertension.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.