Patent · US Expired

Pyridine derivatives

US5075303A · kind A · utility

10Cited by
2References
10Claims
0Family size

Assignee

Inventors

Key dates

Filing dateApr 6, 1990
Grant dateDec 24, 1991
Priority date
Expiry dateApr 6, 2010

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D405/12
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Pyridine derivatives of formula ##STR1## their heteroaromatic N-oxides and their pharmaceutically acceptable acid addition salts are disclosed. In the formula z is 0, 1 and 2 and R, R.sup.1, R.sup.2 and R.sup.2 have specified meanings. The compounds exhibit activity as 5-HT.sub.1A agonists, antagonists or partial agonists and are useful for the treatment of CNS disorders e.g. anxiety, as antihypertensives and in treating anorexia.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.