Guanidinobenzoic ester derivative
US5075335A · kind A · utility
1Cited by
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11Claims
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Key dates
| Filing date | Mar 16, 1990 |
| Grant date | Dec 24, 1991 |
| Priority date | — |
| Expiry date | Mar 16, 2010 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D263/44
- WIPO fieldOrganic fine chemistry
- WIPO sectorChemistry
Abstract
A guanidinobenzoic ester derivative having the formula is novel and effective to inhibit enzymes such as trypsin, plasmin and thrombin, being useful for treatment of the pancreatitis and hemorrhagic disease and thrombosis. ##STR1## wherein X represents a group of the formula: ##STR2## in which Y is a group of the formula: --(CH.sub.2).sub.m --, m being an integer of 2 or 3, ##STR3## or a group of the formula: EQU --OR in which R is a hydrogen atom or a lower alkyl group, and n represents an integer of 1 to 5.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.