Patent · US Expired

1,2,3-triazole compounds active as inhibitors of the enzyme HMG-CoA reductase and pharmaceutical compositions containing them

US5081136A · kind A · utility

17Cited by
1References
7Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 13, 1990
Grant dateJan 14, 1992
Priority date
Expiry dateDec 13, 2010

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D405/06
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Compounds of formula ##STR1## wherein R, R.sub.1, R.sub.2, R.sub.3 and Z have the meanings reported in the specification, and intermediates for their preparation are described. The compounds of formula I have antiatherosclerotic activity as inhibitors of the enzyme HMG-CoA reductase and they are useful in the pharmaceutical field. Compositions for pharmaceutical use containing a compound of formula I as active ingredient are described too.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.