Patent · US Expired

1-aminomethyl-1,2,3,4-tetrahydronaphthalenes

US5086074A · kind A · utility

2Cited by
1References
5Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMar 26, 1990
Grant dateFeb 4, 1992
Priority date
Expiry dateMar 26, 2010

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07C2602/10
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Compounds of the formula ##STR1## and pharmaceutically acceptable salt thereof, wherein R.sup.2 is selected from hydroxy and lower alkoxy, R.sup.5 is lower alkyl, and R.sup.11 and R.sup.12 are independently selected from hydrogen, halo, hydroxy, methoxy, and lower alkyl, are selective .alpha..sub.2 adrenergic receptor antagonists useful in the treatment of glaucoma.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.