Patent · US Expired

6-substituted mitomycin analogs

US5098926A · kind A · utility

0Cited by
11References
24Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 13, 1989
Grant dateMar 24, 1992
Priority date
Expiry dateDec 13, 2009

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D487/14
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Novel methods for treatment of neoplastic disease states in animals, which methods comprise administering a therapeutically effective amount of a compound of the formula IV, ##STR1## wherein: Y is hydrogen or lower alkyl; and X is a radical of the formula --O--R, wherein R is: PA1 a substituted lower alkyl radical selected from the group consisting of mono- and di-hydroxy lower alkyl, cyano lower alkyl, halo lower alkyl, lower alkyl amino lower alkyl, hydroxy lower alkylthio lower alkyl, hydroxy lower alkyldithio lower alkyl, di-lower alkoxy lower alkyl, hydroxy or lower alkoxy substituted lower alkoxy lower alkyl, cyclo lower alkyl substituted lower alkyl; and lower alkyl substituted dioxolanyl lower alkyl or PA1 a lower alkenyl radical; or PA1 a lower alkynyl radical; or PA1 tetrahydro furanyl or a lower alkyl substituted derivative thereof, oxiranyl lower alkyl, tetrahydropyranyl lower alkyl, or furanyl lower alkyl.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.