Patent · US Expired

Novel sulfonylphenyl-.beta.-D-thioxylosides, their method of preparation and their use in therapeutics

US5100913A · kind A · utility

4Cited by
1References
8Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMar 25, 1991
Grant dateMar 31, 1992
Priority date
Expiry dateMar 25, 2011

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07C323/65
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention relates, by way of novel industrial products, to the sulfonylphenyl-.beta.-D-thioxyloside compounds of the formula ##STR1## in which: X is a sulfur atom or an oxygen atom; PA1 R is a C.sub.1 -C.sub.4 alkyl group, a substituted amino group NR.sub.1 R.sub.2 (where R.sub.1 and R.sub.2, which are identical or different, are each a C.sub.1 -C.sub.4 alkyl group, it being possible for R.sub.1 and R.sub.2, taken together, to form a piperidinyl or morpholinyl group with the nitrogen atom to which they are bonded) or a phenyl group which is unsubstituted or substituted in the para position by a cyano group or by a halogen atom; and PA1 Y is the hydrogen atom or an aliphatic acyl group. These compounds are useful in therapeutics, especially as venous antithrombotics.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.