Patent · US Expired

2,9-dihydro-(6 or 7)-(3-oxo-2,3,4,5-tetrahydropyridazinyl)-pyrazolo [4,3-B]-1,4-benzoxazines

US5116837A · kind A · utility

3Cited by
5References
9Claims
0Family size

Assignee

Inventor

Key dates

Filing dateDec 21, 1990
Grant dateMay 26, 1992
Priority date
Expiry dateDec 21, 2010

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P9/08
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The invention relates to novel compounds, 2,9-dihydro(6 or 7)-3-oxo-2,3,4,5-tetrahydropyridazinyl)pyrazolo[4,3-b]benzoxazines. The claimed compounds are inhibitors of phosphodiesterase fraction III and have potent positive inotropic activity. These compounds are useful as cardiotonics or platelet aggregation inhibitors. This invention also pertains to compositions comprising an effective amount of the compounds, to methods for preparing the claimed compounds and to methods for treating a mammal with the compounds.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.