Patent · US Expired

Platelet activating antagonists

US5120749A · kind A · utility

5Cited by
3References
8Claims
0Family size

Assignee

Inventors

Key dates

Filing dateFeb 20, 1991
Grant dateJun 9, 1992
Priority date
Expiry dateFeb 20, 2011

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D417/14
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Indole compounds substituted at the 1- or 3 position by a (pyrid-3 yl)thiazolid-4-yl)alkyl-, (pyrid-3-yl)thiazolid-4-oyl)-, (pyrid-3-yl)dithiolan-4-yl)alkyl- or (pyrid-3-yl) dithiolan-4-ol)- group are potent inhibitors of PAF and are useful in the treatment of PAF-related disorders including anaphylactic shock, respiratory distress syndrome, acute inflammation, delayed cellular immunity, parturtition, fetal lung maturation, and cellular differentiation.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.