Patent · US Expired

Benzoxazolinone compounds, compositions and use

US5132305A · kind A · utility

10Cited by
1References
10Claims
0Family size

Assignee

Inventors

Key dates

Filing dateFeb 26, 1990
Grant dateJul 21, 1992
Priority date
Expiry dateFeb 26, 2010

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D417/06
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Compounds of general formula (I): ##STR1## in which: R.sub.1 denotes a hydrogen atom or a lower alkyl optionally substituted with a hydroxyl group, PA0 R.sub.2 and R.sub.3 : PA1 a--identical or different, denote a hydrogen atom, a lower alkyl, a lower alkenyl, a substituted or unsubstituted aryl, a substituted or unsubstituted (lower alkyl)aryl, PA1 b--are such that they form, with the nitrogen which carries them, a saturated or unsaturated, mono- or bicyclic heterocyclic system containing at most 3 hetero atoms per ring, substituted or unsubstituted, with the exception of 1-arylpiperazine systems, PA0 X denotes a hydrogen atom, PA0 Y denotes a hydrogen atom or a hydroxyl, or alternatively X and Y denote an oxygen atom, provided that R.sub.1 is then other than a methyl group, PA0 Z denotes a hydrogen atom or forms a .pi. bond with Y, and PA0 T denotes a hydrogen atom or a lower alkyl, their stereoisomers and their quaternary ammonium salts, as well as their addition salts with a pharmaceutically acceptable acid.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.