Heterocyclic acetylenic amines having central nervous system activity
US5137905A · kind A · utility
2Cited by
4References
4Claims
0Family size
Assignee
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Key dates
| Filing date | Apr 5, 1991 |
| Grant date | Aug 11, 1992 |
| Priority date | — |
| Expiry date | Apr 5, 2011 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D249/08
- WIPO fieldOrganic fine chemistry
- WIPO sectorChemistry
Abstract
Heterocyclic acetylenic amine compounds having the following structural formula ##STR1## having cholinergic agonist or antagonist activity useful in the treatment of mental disorders, extrapyramidal motor disorders, disorders of the parasympathetic nervous system and glaucoma or as analgesics for the treatment of pain. Typical central nervous system disorders for which the subject compounds can be used include cognitive disorders of all ages, including senile dementia, Alzheimer's disease and other related disorders. The compounds are particularly developed to improve mental performance when a mental deficiency is diagnosed.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.