Patent · US Expired

Phosphonate, phosphinate derivatives useful as antihypertensive agents

US5153347A · kind A · utility

25Cited by
10References
5Claims
0Family size

Assignee

Inventor

Key dates

Filing dateJan 31, 1991
Grant dateOct 6, 1992
Priority date
Expiry dateJan 31, 2011

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07F9/4075
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Novel angiotensin II receptor antagonists of the formula ##STR1## wherein X, X.sub.1, X.sub.2, R.sub.1, R.sub.2, R.sub.3, R.sub.4 and R.sub.5 are as defined herein, are disclosed. These compounds are useful, for example, in the treatment of hypertension, congestive heart failure and cardiac hypertrophy.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.