Patent · US Expired

Preparation of 2-alkylthio-1,3,4-thiadiazoles

US5162539A · kind A · utility

5Cited by
4References
9Claims
0Family size

Assignee

Inventor

Key dates

Filing dateJan 25, 1991
Grant dateNov 10, 1992
Priority date
Expiry dateJan 25, 2011

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D285/125
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

A process for the preparation of a 2-alkylthio-1,3,4-thiadiazole of the formula ##STR1## in which R.sup.1 represents alkyl which is optionally substituted by halogen and PA0 R.sup.2 represents alkyl or aralkyl, which comprises reacting a carboxylic acid of the formula EQU R.sup.1 --COOH (II), with a dithiocarbazic ester of the formula ##STR2## in the presence of phosphoryl chloride (POCl.sub.3) at a temperature between -20.degree. C. and +120.degree. C.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.