Patent · US Expired

4(3H)-pteridinones, preparation processes and drugs containing them

US5167949A · kind A · utility

35Cited by
9References
20Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMar 29, 1990
Grant dateDec 1, 1992
Priority date
Expiry dateMar 29, 2010

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P37/08
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention relates to 4(3H)-pteridinones represented by the formula: ##STR1## in which X is an oxygen atom or a sulphur atom, Y is a hydrogen atom, a lower alkyl radical, especially a methyl radical, at the 6-position or a hydroxyl group at the 7-position, R.sub.1 is a hydrogen atom, a lower alkyl radical, a substituted or unsubstituted phenyl radical, a benzyl radical, a methoxymethyl group, an acetyl group, a 2-acetoxyethyl group or a 2,2,2-trifluoroethyl group and R.sub.2 is a hydrogen atom or a lower alkyl radical, especially a methyl radical. Application of these compounds as anti-allergic drugs.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.