Benzisoxazole and benzisothiazole compounds
US5173490A · kind A · utility
6Cited by
9References
13Claims
0Family size
Assignee
Inventors
Key dates
| Filing date | Jan 7, 1992 |
| Grant date | Dec 22, 1992 |
| Priority date | — |
| Expiry date | Jan 7, 2012 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D261/20
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
The compounds are N-substituted N'-(benzisoxazolyl or benzisothiazolyl) piperazines useful as sedative, anxiolytic, anti-aggressive and analgesic agents and for the treatment of schizophrenia and depression. A compound disclosed is (R,S)-3-{1-[(benzocyclobutan-1-yl)methyl]piperazin-4-yl}-6-fluoro-1,2-benz isoxazole.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.