Patent · US Expired

Serotonergic alpha-oxoacetamides

US5192770A · kind A · utility

38Cited by
3References
34Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 7, 1990
Grant dateMar 9, 1993
Priority date
Expiry dateDec 7, 2010

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D487/08
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

.alpha.-Oxoacetamides of the formula R.sup.1 C(O)C(O)NR.sup.2 R.sup.3 in which R.sup.1 is optionally substituted phenyl, 1-indolyl, 2,3-dihydro-1-indolyl, 1-benzimidazolidinonyl, 3-benzofuranyl, 3-benzothiophenyl, 3-indolyl, and 1,2-alkano-3-indolyl; R.sup.2 is selected from: ##STR1## and R.sup.3 is selected from hydrogen or lower alkyl; and the pharmaceutically acceptable salts, individual isomers, mixtures of isomers, processes for preparation, compositions, and methods of use thereof.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.