Patent · US Expired

Method for enhancing the safety of metal-ligand chelates as X-ray contrast agents

US5204085A · kind A · utility

11Cited by
6References
13Claims
0Family size

Assignee

Inventor

Key dates

Filing dateNov 18, 1991
Grant dateApr 20, 1993
Priority date
Expiry dateNov 18, 2011

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K49/06
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Paramagnetic chelates, as for example, Gadolinium diethylenetriaminepentaacetic acid (DTPA), manganese, ethylenediaminetetraacetic acid (EDTA), and others used as X-ray contrast agents are more toxic acutely when injected in high concentration or at rapid rates. The use of effective amounts of calcium in the form of, calcium chloride, calcium gluconate, or balanced salt solutions substantially reduces this toxicity without the need to add additional ligand.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.